Preclinical assessment of a novel small molecule inhibitor of tryptophan 2,3-dioxygenase 2 (TDO2)

نویسندگان

  • Stefano Crosignani
  • Gregory Driessens
  • Michel Detheux
  • Benoît Van den Eynde
  • Sandra Cauwenberghs
چکیده

Introduction iTeos leverages the science of LICR to target metabolism of the tumor microenvironment and develops small molecule immunomodulators. TDO2 is a heme-containing enzyme highly expressed in the liver, in specific brain regions and liver/brain tumors. It catalyses the first and rate-limiting step of tryptophan catabolism along the kynurenine pathway and thereby regulates systemic tryptophan levels. Tryptophan (Trp) degradation by TDO2 suppresses anti-tumor immune responses and promotes tumor cell survival.

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عنوان ژورنال:

دوره 2  شماره 

صفحات  -

تاریخ انتشار 2014